R. Karmakar, A. Rheingold, G. C. Micalizio, “Studies Targeting Ryanodol Result in an Annulation Reaction for the Synthesis of a Variety of Fused Carbocycles” Org. Lett. 2019, 21, 6126-6129.
R. M. Leon, D. Ravi, J. S. An, C. L. del Genio, A. Rheingold, A. B. Gaur, G. C. Micalizio, “Synthesis of C14-Desmethylene Corialactone D and the Discovery of Inhibitors of Nerve Growth Factor-Mediated Neurite Outgrowth” Org. Lett. 2019, 21, 3193-3197.
W. S. Kim, Z. A. Shalit, S. Nguyen, E. Schoepke, A. Eastman, T. P. Burris, A. B. Gaur, G. C. Micalizio, “A Synthesis Strategy for Tetracyclic Terpenoids Leads to Agonists of ERb” Nature Commun. 2019, 10, article #2448 (DOI: 10.1038/s41467-019-10415-6).
A. B. Millham, M. J. Kier, R. M. Leon, R. Karmakar, Z. D. Stempel, G. C. Micalizio, “A Complementary Process to Pauson–Khand-type Annulation Reactions for the Construction of Fully Substituted Cyclopentenones” Org. Lett. 2019, 21, 567-570.
K. Du, M. J. Kier, A. Rheingold, G. C. Micalizio, “Toward the Total Synthesis of Ryanodol via Oxidative Alkyne–1,3-Diketone Annulation: Construction of a Ryanoid Tetracycle” Org. Lett. 2018, 20, 6457-6461.
W. S. Kim, K. Du, A. Eastman, R. P. Hughes, G. C. Micalizio “Synthetic nat- or ent-steroids in as few as five chemical steps from epichlorohydrin” Nat. Chem. 2018, 10, 70-77.
N. F. O’Rourke, G. C. Micalizio “Function-Oriented Studies Targeting Pectenotoxin 2: Synthesis of the GH-Ring System and a Structurally Simplified Macrolactone” Org. Lett. 2017, 19, 5154-5157.
M. J. Kier, R. M. Leon, N. F. O’Rourke, G. C. Micalizio “Synthesis of Highly Oxygenated Carbocycles by Stereoselective Coupling of Alkynes to 1,3- and 14,-Dicarbonyl Systems” J. Am. Chem. Soc. 2017, 139,12374-12377.
W. S. Kim, K. Du, R. P. Hughes, G. C. Micalizio “Synthetic nat- or ent- steroids in as few as five chemical steps from epichlorohydrin” Nat. Chem. 2017, 9, DOI: 10.1038/nchem.2865.
H. Mizoguchi, G. C. Micalizio “Convergent Synthesis of Angularly Substituted Trans-Decalins by a Metallacycle-mediated Cross-Coupling Reaction Cascade” Angew. Chem. Int. Ed. 2016, accepted.
G. C. Micalizio, N. F. O’Rourke, M. J. Kier “Metallacycle-mediated Cross-Coupling in Natural Product Synthesis” invited Report – Tetrahedron, 2016, accepted.
C. Aquino, S. N. Greszler, G. C. Micalizio “Access to the Cortistatin Pentacyclic Core by Alkoxide-Directed Metallacycle-Mediated Annulative Cross-Coupling” Org. Lett. 2016, 18, 2624-2627.
N. F. O'Rourke, G. C. Micalizio, "Cyclopropenes in Metallacycle-Mediated Cross-Coupling with Alkynes: Convergent synthesis of highly substituted vinylcyclopropanes" Org. Lett. 2016, 18, 1250-1253.
X. Cheng, G. C. Micalizio, "Synthesis of Neurotrophic Seco-prezizaane Sesquiterpenes (1R,10S)-2-oxo-3,4-dehydroneomajucin, (2S)-hydroxy-3,4-dehydroneomajucin, and (–)-jiadifenin" J. Am. Chem. Soc. 2016, 138, 1150-1153.
H. Mizoguchi, G. C. Micalizio “Synthesis of Highly Functionalized Decalins via Metallacycle-Mediated Cross-Coupling” J. Am. Chem. Soc. 2015, 137, 6624-6628.
X. Cheng, G. C. Micalizio “An Annulation Reaction for the Synthesis of Cross-Conjugated Triene-containing Hydroindanes from Acyclic Precursors” Org. Lett. 2014, 16, 5144-5147.
V. Jeso, C. Aquino, X. Cheng, H. Mizoguchi, M. Nakashige, G. C. Micalizio, “Direct Synthesis of Angularly Substituted Trans-fused Hydroindanes by Convergent Coupling of Acyclic Precursors” J. Am. Chem. Soc. 2014, 136, 8209-8212.
V. Jeso, S. Iqbal, P. Hernandez, M. D. Cameron, H. Park, P. V. LoGrasso, G. C. Micalizio “Synthesis of Benzoquinone Ansamycin-Inspired Macrocyclic Lactams from Shikimic Acid” Angew. Chem. Int. Ed. 2013, 52, 4800-4804.
D. Yang, G. C. Micalizio “Synthesis of Alkaloid (–)-205B via Stereoselective Reductive Cross-Coupling and Intramolecular [3+2] Cycloaddition” J. Am. Chem. Soc. 2012, 134, 15237-15240.
S. Greszler, H. A. Reichard, G. C. Micalizio, “Asymmetric Synthesis of Dihydroindanes by Convergent Alkoxide-Directed Metallacycle-Mediated Bond Formation” J. Am. Chem. Soc. 2012, 134, 2766-2774.
M. Z. Chen, G. C. Micalizio “Three-Component Coupling Sequence for the Regiospecific Synthesis of Substituted Pyridines” J. Am. Chem. Soc. 2012, 134, 1352-1356.
C. Aquino, M. Sarkar, M. J. Chalmers, K. Mendez, T. Kodadek, G. C. Micalizio “A Biomimetic Polyketide-Inspired Approach to Small Molecule Ligand Discovery” Nature Chem. 2012, 4, 99-104.
D. Yang, G. C. Micalizio, “Convergent and Stereodivergent Synthesis of Complex 1-Aza-7-Oxabicyclo[2.2.1]heptanes” J. Am. Chem. Soc. 2011, 133, 9216-9219.
M. A. Tarselli, K. M. Raehal, A. K. Brasher, C. Groer, M. D. Cameron, L. M. Bohn, G. C. Micalizio, “Synthesis of Conolidine, a Potent Non-Opioid Analgesic for Tonic and Persistent Pain” Nature Chem. 2011, 3, 449-453.
V. Jeso, G. C. Micalizio, “Total Synthesis of Lehualide B by Allylic Alcohol–Alkyne Reductive Cross-Coupling” J. Am. Chem. Soc. 2010, 132, 11422-11424.
D. P. Canterbury, G. C. Micalizio, “Polyketide Assembly by Alkene–Alkyne Reductive Cross-Coupling: Spiroketals Through the Union of Homoallylic Alcohols” J. Am. Chem. Soc. 2010, 132, 7602-7604.
T. K. Macklin, G. C. Micalizio, “Convergent and Stereospecific Synthesis of Skipped Polyenes and Polyunsaturated Fatty Acids” Nature Chem. 2010, 2, 638-643.
D. Yang, G. G. Micalizio, “A Convergent Stereoselective Synthesis of Quinolizidines and Indolizidines: Chemoselective Coupling of 2-Hydroxymethyl Substituted Allylic Silanes with Imines” J. Am. Chem. Soc. 2009, 131, 17548-17549.